13
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T60872 | Adenosine receptor antagonist 3 | ||
Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1]. | |||
T21389 | Enprofylline | Enprofilina,3-propylxanthine,3-n-Propylxanthine,Enprofyllinum | Others |
Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor. Enprofylline is used in asthma, chronic obstructive pulmonary disease, and in the management of sick... | |||
T68132L | Quercetin-3'-o-phosphate TEA | Quercetin-3'-o-phosphate TEA(1111616-69-3 Free base),3'-quercetin phosphate TEA,Quercetin 3'-phosphate TEA | Adenosine Receptor |
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders. | |||
T6552 | Istradefylline | KW-6002 | Adenosine Receptor |
Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails. It has been used in trials studying the treatment and basic science of Drug Ab... | |||
T62611 | Adenosine receptor antagonist 2 | ||
Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects. | |||
T25841 | MSX-3 | MSX 3 | |
MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2. | |||
T69566 | MSX-3 free acid | ||
MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2. | |||
T62797 | A2A receptor antagonist 3 | ||
A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM). | |||
T62134 | A1/A3 AR antagonist 1 | ||
A1/A3 AR antagonist 1 (Compound 10) is a potent, dual adenosine 1 (A1) and adenosine 3 (A3) receptor antagonist that acts on human A1 (Ki: 37.6 nM), human A3 (Ki: 25.4 nM) and rat A1 (Ki: 1.47 nM). 1 Can be used to study... | |||
T72626 | A2AR-antagonist-1 | Adenosine Receptor | |
A2AR-antagonist-1 (compound 38), an orally active adenosine A2A receptor antagonist with an IC50 value of 29 nM, demonstrates anti-tumor properties and stability in mouse liver microsomes (t1/2 = 86.1 min). Additionally,... | |||
T71328 | Theobromine-d6 | ||
Theobromine-d6 is intended for use as an internal standard for the quantification of theobromine by GC- or LC-MS. Theobromine is a methylxanthine alkaloid and derivative of caffeine that has been found in cocoa beans and... | |||
T60511 | Theophylline sodium glycinate | ||
Theophylline (1,3-Dimethylxanthine) sodium glycinate is a potent inhibitor of phosphodiesterase (PDE) that inhibits PDE3 activity to relax airway smooth muscle. Theophylline sodium glycinate can be used for the research ... | |||
T36679 | Rp-cAMPS sodium salt | ||
Rp-cAMPS sodium salt, a cAMP analog, is a potent, competitive cAMP-induced activation of cAMP-dependent PKA I and II (Kis of 12.5 μM and 4.5 μM, respectively) antagonist. Rp-cAMPS sodium salt is resistant to hydrolysis b... |